Exemestane - a drug which is the same as Letrozole or Anastrozole, aromatase inhibitors. It is used to reduce the concentration of estrogen in the blood and increase own male testosterone hormone levels. And so also for preventing or treating gynecomastia in men.
Exemestane - a new generation of drug that blocks enzymes responsible for aromatisation. Exemestane is called a true aromatase killer. The principle of action of this drug is that it blocks enzymes responsible for the synthesis of estrogens.
Many experienced athletes believe that Exemestane is the most effective aromatase inhibitor. This drug inhibits at least 85% of estrogens. And it should be noted that it is a suppression of an irreversible process. Of course, there are many other highly effective drugs, but if you read on AROMASIN (Exemestane) reviews, you can make sure that athletes give preference to the drug because of its high efficiency in combating gynecomastia, fat accumulation and fluid in the body.
The drug was made in 1999 year. The purpose of its invention - the treatment of breast cancer disease. Bodybuilders use it during the cycle of a steroid with a large percentage of flavoring. Exemestane action is radically different from that of the same Tamoxifen, which does not affect the process of flavoring, it simply does not join the estrogen and estrogen receptors form a bond. But the effect of Exemestane is aimed at suppressing the flavoring process.
Exemestane is significantly different from their counterparts, drugs aromatase inhibitors, it is more refined. The effect of taking this drug is irreversible and permanent, while other aromatase inhibitors have a temporary effect.
Aromasin side effects include: fatigue, depression, pain in the head, rash, excessive sweating. The manifestation of the side effects of the drug is purely individual. Depending on the sensitivity of the body to the drug. Often, the cost of the drug is rather high, but its efficient and operational without doubt.
Exemestane Cycle / Dosage
The amount required of Exemestane is calculated taking into account the use of anabolic steroids, individual sensitivity to aromatase inhibitors. In the most general case, Exemestane dosage equals to 12.5 mg per day. It should be remembered that the use of Exemestane is only necessary to control the levels of estrogen. Full reduction or removal of estrogen has a negative impact on the body.
The duration of the drug is 2-4 weeks. In the event that an athlete has not started in time to take aromatase inhibitors and are already visible or pronounced estrogenic side effects, you should start taking Exemestane 25 mg daily and do not stop taking the drug until the complete disappearance of symptoms of gynecomastia.
It is recommended to take Exemestane during meals or immediately after it. In this case, bioavailability will increase by 40%, and two hours later will be reached its maximum concentration in blood.